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Rational Engineering of Isoform-Specific Hsult1e1 Fluorogenic Substrates for Functional Analysis and Inhibitor Screening

Xiaoting Niu,Yufan Fan, Guanghao Zhu,Hairong Zeng,Bei Zhao, Mengru Sun, Lin Chen,Luling Wu,Zhenhao Tian,Tony D. James,Guangbo Ge

Biosensors and Bioelectronics(2025)

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关键词
human estrogen sulfotransferase (hSULT1E1),structure-based substrate design,enzyme activity analysis,high-throughput screening
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