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Discovery and Exploration of Disubstituted [1,2,5]Oxadiazolo-[3,4-b]pyrazines As Novel C-C Chemokine Receptor Type 5 Signaling Inhibitors Targeting the Intracellular Allosteric Binding Pocket

Margaux Billen, Sten Reynders,Sandra Claes, Silke Kleinboelting, Jef Rozenski, Radu-George Bulai, Edoardo Rocca,Natalie Z M Homer,Scott P Webster, Tim P Kaminski,Eveline Lescrinier,Dominique Schols,Peter Verwilst

European journal of medicinal chemistry(2025)

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