KT-253, A Novel MDM2 Degrader and P53 Stabilizer, Has Superior Potency and Efficacy Than MDM2 Small Molecule Inhibitors
Yogesh K Chutake, Michele F Mayo, Nancy Dumont,Jessica Filiatrault, Susanne B Breitkopf,Patricia Cho,Dapeng Chen, Vaishali S Dixit, William R Proctor, Eric W Kuhn, Sarah Bollinger Martinez,Alice A McDonald, Jianfeng Qi,Kan-Nian Hu,Rahul Karnik,Joseph D Growney,Kirti Sharma,Stefanie S Schalm, Ashwin M Gollerkeri,Nello Mainolfi, Juliet A Williams,Matthew M Weiss Molecular cancer therapeutics(2025)
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