Discovery of A-910, a Highly Potent and Orally Bioavailable Dual MerTK/Axl-Selective Tyrosine Kinase Inhibitor.
Yiyun Yu,Miyeon Jang, Julie Miyashiro,Richard F. Clark,Gui-Dong Zhu,Jane Gong,Yujia Dai,Robin R. Frey,Thomas D. Penning, Hadong Kim,Hyung Ki Lee, Jin Kwan Kim,Ki Moon Ryu, Seong Jin Park,Taeyoung Yoon, Tao Li, Matthew D. Kurnick, Nicolas J. Kapecki,Leiming Li, Jacob V. Gorman,Debra A. Montgomery,Vlasios Manaves,Kenneth D. Bromberg,Stella Z. Doktor, Ashish Thakur,Jin Wang, Heath A. Smith,Fritz G. Buchanan,Debra C. Ferguson,Maricel Torrent,Clarissa G. Jakob,Wei Qiu,Anup K. Upadhyay,Ruth L. Martin,Albert Lai,Michael R. Michaelides JOURNAL OF MEDICINAL CHEMISTRY(2024)
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