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Development of a Scalable Alkylation Via a Protection/Deprotection Sequence for BMT-773752: Key Intermediate in the Synthetic Route to Repotrectinib

Han Zhang, Binfeng Li, Jin Yang, Changchun Xu,Rafaela Carmona,Jason Zhu, Bilal Hoblos,Steven Wisniewski

Organic Process Research & Development(2024)

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关键词
starting material,alkylation,salt formation,crystallization
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