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Development of a Safe and Scalable Method to Prepare 3-Bromo-n-alkyl-1,6-naphthyridones Via Enamine Cyclization

Thomas Carr, Sam Beddoe, Stephen Johns, Jonathan Hull, Tom Stowe, Jonathan Moore, James Brown, Adrian Maddaford,Etienne Rochette,Michel Bernatchez, Martin Jean, Jean Francois Parent, Connor Barrett,Jeffrey B. Sperry, Daniel Richter

ORGANIC PROCESS RESEARCH & DEVELOPMENT(2024)

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关键词
enamine,naphthyridone,cyclization,annulation
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