Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models (vol 62, pg 6540, 2019) M. Raymond V. Finlay , Mark Anderton , Andrew Bailey , Scott Boyd , Joanna Brookfield , Ceri Cairnduff , Mark Charles , Anne Cheasty , Susan E. Critchlow , Janet Culshaw , Judit Debreczeni , Tennyson Ekwuru , Ian Hollingsworth , Neil Jones , Fred Leroux , Mairi Littleson , Hollie McCarron , Jennifer McKelvie , Lorraine Mooney , J. Willem M. Nissink , Joe Patel , David Perkins , Steve Powell , Mar Jimenez Quesada , Piotr Raubo , Verity Sabin , James Smith , Peter D. Smith , Andrew Stark , Attilla Ting , Peng Wang , Zena Wilson , Jon J. Winter-Holt , J. Matthew Wood , Gail L. Wrigley , Guoqing Yu , Peng Zhang JOURNAL OF MEDICINAL CHEMISTRY(2023)
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