Process Development of the BACE Inhibitors BI 1147560 BS and BI 1181181 MZ
Guisheng Li,Zhulin Tan,Yibo Xu,Kanwar P. S. Sidhu,Bo Qu,Melissa A. Herbage,Magnus C. Eriksson,Xingzhong Zeng,Carl A. Busacca,Jean-Nicolas Desrosiers, Thomas Hampel,Oliver Niemeier, Carsten Reichel, Mai Thi Quynh Dang, Marvin Schoerer,Dirk Kemmer, Melanie Eick, Holger Werle,Soojin Kim,Zhibin Li,Shankar Venkatraman,Lanqi Jia,David A. Claremon,Klaus Fuchs,Niklas Heine,Denis Byrne,Bikshandarkoil Narayanan,Max Sarvestani,Joe Johnson,Ajith Premasiri,Larry J. Nummy,Jon C. Lorenz,Nizar Haddad,Nina C. Gonnella,Scott Pennino,Mariusz Krawiec,Chris H. Senanayake,Frederic Buono,Heewon Lee,Azad Hossain,Jinhua J. Song,Jonathan T. Reeves Organic process research & development(2022)
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carbamoyl anion,transnitrilation,oxetane,fluorination
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