Discovery of the First Selective Nanomolar Inhibitors of Endoplasmic Reticulum Aminopeptidase 2 by Kinetic Target‐Guided Synthesis
Virgyl Camberlein, Charlotte Fleau-Tabey,Pierre Sierocki,Lenong Li,Ronan Gealageas,Damien Bosc,Valentin Guillaume,Sandrine Warenghem,Florence Leroux,Melissa Rosell,Keguang Cheng,Laura Medve,Mathilde Prigent,Myriam Decanter,Catherine Piveteau,Alexandre Biela,Maxime Eveque,Julie Dumont,Anastasia Mpakali,Petros Giastas,Adrien Herledan,Cyril Couturier,Jörg Haupenthal,Laetitia Lesire,Anna K Hirsch,Benoit Deprez,Efstratios Stratikos,Marlene Bouvier,Rebecca Deprez-Poulain Angewandte Chemie International Edition(2022)
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