Synthesis of Way-163909; a Selective 5-Ht2cr Agonist
SSRN Electronic Journal(2022)
摘要
A new synthetic approach to derivatives the serotonin 2C receptor (5-HT2CR) agonist WAY-163909 is reported. In addition to the WAY-163909 versions possessing a site that has been shown to accommodate the attachment of linkers without loss of agonist activity are accessible by this approach. An efficient 7 step synthesis with an overall 32% yield is reported.
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关键词
Serotonin,Benzodiazepine,N-heteroannulation,WAY-163909,5-HT2C,5-HT2CR
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