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Manufacturing Process Development for Belzutifan, Part 1: A Concise Synthesis of the Indanone Starting Material

Feng Peng,Lushi Tan,Lu Chen,Stephen M. Dalby,Daniel A. DiRocco,Jianjun Duan, Minyi Feng, Guan Gong, Haiheng Guo,J. Caleb Hethcox, Lu Jin,Heather C. Johnson,Jungchul Kim,Diane Le,Yipeng Lin,Wenjun Liu, Jun Shen, Yimei Wan,Chengqian Xiao,Bangping Xiang, Qun Xiang, Jing Xu, Luliang Yan, Weiyi Yang,Honglin Ye, Yanpei Yu, Jun Zhang

Organic Process Research & Development(2021)

Cited 25|Views4
Key words
belzutifan,Friedel-Crafts cyclization,CuBr-promoted sulfonylation
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