Discovery Of A Novel Class Of Potent, Selective, And Orally Bioavailable Histone Methyltransferase Enhancer Of Zeste Homolog 2 (Ezh2) Inhibitors And The Identification Of Development Candidate Pf-06821497 Pei-Pei Kung , Simon Bergqvist , Patrick Bingham , John Braganza , Alexei Brooun , Michael Collins , Wade Diehl , Ya-Li Deng , Dac Dinh , Connie Fan , Valeria Fantin , Hovhannes Gukasyan , Wenyue Hu , Buwen Huang , Robert Kania , Wei Liu , Susan Kephart , Manfred Kraus , Cody Krivacic , Robert Kumpf , Gary Li , Karen Maegley , Indrawan Mcalpine , Lisa Nguyen , Sacha Ninkovic , Martha Ornelas , Dan Richter , Eugene Rui , Michael Ryskin , Stephanie Scales , Jillian Spangler , Al Stewart , Scott Sutton , John Tatlock , Cheng-Chung Tsao , Dominique Verhelle , Fen Wang , Hui Wang , Peter Wells , Martin Wythes , Shinji Yamazaki , Brian Yip , Xiu Yu , Luke Zehnder , Wei-Guo Zhang , Peter Zhu , Jinjiang Zhu , Robert Rollins , Shikhar Sharma , Martin Edwards ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY(2017)
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