Discovery of a Series of 7-Azaindoles As Potent and Highly Selective CDK9 Inhibitors for Transient Target Engagement.
Bernard Barlaam,Chris De Savi,Allan Dishington,Lisa Drew,Andrew D. Ferguson,Douglas Ferguson,Chungang Gu,Sudhir Hande,Lorraine Hassall,Janet Hawkins,Alexander W. Hird,Jane Holmes,Michelle L. Lamb,Andrew S. Lister,Thomas M. McGuire,Jane E. Moore,Nichole O'Connell,Anil Patel,Kurt G. Pike,Ujjal Sarkar,Wenlin Shao,Darren Stead,Jeffrey G. Varnes,Melissa M. Vasbinder,Lei Wang,Liangwei Wu,Lin Xue,Bin Yang,Tieguang Yao Journal of Medicinal Chemistry(2021)
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