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欧前胡素与异欧前胡素同牛血清白蛋白相互作用研究?

Yujie ZHANG, Shanshan FAN, Yupei ZHANG

wf(2017)

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Abstract
建立测定欧前胡素与异欧前胡素和牛血清白蛋白(BSA)结合率的高效液相色谱的方法,为临床合理用药提供依据.采用平衡透析-高效液相色谱法测定欧前胡素与异欧前胡素与 BSA 的蛋白结合率.欧前胡素与牛血清白蛋白的结合率为79.3%,异欧前胡素与牛血清白蛋白的结合率为72.7%.在体外欧前胡素和异欧前胡素和牛血清白蛋白结合性较高,且蛋白结合率随着含药白蛋白浓度的增加无明显的浓度依赖性.
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