Rhodium-catalyzed direct CH amination of 2-arylindoles and 7-arylindoles with free amines
TETRAHEDRON LETTERS(2021)
摘要
•NH-indole-directed CH cleavage.•Mild reaction conditions.•High functional group tolerability.•32 examples, up to 95% yield.
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关键词
Rhodium-catalyzed,2-Arylindoles,7-Arylindoles,CH amination,Free amine
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