The Putative KCC2 Activating Small Molecule CLP257 Does not Have any Target Engagement or Functional Activity at KCC2 but Does Potentiates GABAA Receptor Activity

Ross Cardarelli,Karen Jones, Lucie Pisella,Lisa McWilliams, David Baker,Matthew Burnham,Heike Wobst,Qi Wang, Igor Medyna,Tarek Deeb,Stephen Moss, Nicholas Brandon

NEUROPSYCHOPHARMACOLOGY(2016)

引用 0|浏览4
暂无评分
关键词
kcc2,Drug Discovery - New Approaches,GABAA Receptors,Pharmacology
AI 理解论文
溯源树
样例
生成溯源树,研究论文发展脉络
Chat Paper
正在生成论文摘要