Potent anti-tumor activity correlated with inhibition of DNA damage response genes with highly selective and orally bioavailable CDK12 covalent inhibitors

R. Poddutoori,S. Rajagopalan,S. Mukherjee, S. Marappan, D. Samiulla,S. Nayak, S. Sivakumar,M. Ravindra, S. Gore, A. Dhudashiya, K. Charamanna,G. Daginakatte, S. Chelur,M. Ramachandra, S. Samajdar

EUROPEAN JOURNAL OF CANCER(2018)

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