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Disruption of a Key Ligand-H-bond Network Drives Dissociative Properties in Vamorolone for Duchenne Muscular Dystrophy Treatment.

Xu Liu,Yashuo Wang, Jennifer S. Gutierrez,Jesse M. Damsker, Kanneboyina Nagaraju,Eric P. Hoffman,Eric A. Ortlund

Proceedings of the National Academy of Sciences(2020)

引用 52|浏览24
关键词
glucocorticoid receptor,dissociative agonist,allostery,molecular dynamics,nuclear receptor
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