Discovery and Biological Evaluation of Proteolysis Targeting Chimeras (protacs) As an EGFR Degraders Based on Osimertinib and Lenalidomide.
Bioorganic & Medicinal Chemistry Letters(2020)
关键词
Proteolysis targeting chimera,CRBN,EGFR-TK degrader,Osimertinib,Lenalidomide
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