Optimization of a Binding Fragment Targeting the "enlarged Methionine Pocket" Leads to Potent Trypanosoma Brucei Methionyl-Trna Synthetase Inhibitors.
Bioorganic & Medicinal Chemistry Letters(2017)
关键词
Human African trypanosomiasis,Methionyl-tRNA synthetase,Structure-based design,Trypanosoma brucei
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