Drug Likeness and Selective Functionalization of Quinoxalines

CURRENT ORGANIC SYNTHESIS(2015)

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摘要
In recent years, the pharmacological potential of quinoxalines has received vast interest due to its many applications. This review centers on a critical overview of chemical diversity and physicochemical properties of bioactive quinoxaline libraries. In addition, recent strategies for obtaining structurally diverse quinoxalines using highly selective processes will be discussed.
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关键词
Quinoxaline,heterocycles,C-H activation,drug-likeness,organometallics
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