Discovery of Novel, Potent, Selective and Cellular Active ADC Type PTP1B Inhibitors Via Fragment-Docking-oriented De Novel Design
Bioorganic & Medicinal Chemistry(2015)
关键词
Protein tyrosine phosphatase 1B inhibitor,N-(2,5-Diethoxy-phenyl)-methanesulfonamide,Type 2 diabetes mellitus,Insulin signaling
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