ChemInform Abstract: Indole RSK Inhibitors. Part 2. Optimization of Cell Potency and Kinase Selectivity.
Cheminform(2012)
摘要
A series of inhibitors for the 90 kDa ribosomal S6 kinase (RSK) are optimized for cellular potency and kinase selectivity.
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关键词
indole rsk inhibitors,kinase selectivity,cell potency
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