Synthesis of new N-(arylcyclopropyl)acetamides and N-(arylvinyl)acetamides as conformationally-restricted ligands for melatonin receptors.
Bioorganic & Medicinal Chemistry Letters（2013）
摘要
New constrained analogues of melatonin have been prepared and evaluated on human MT1 and MT2 receptors.
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关键词
Melatonin,MT1 and MT2 receptors,Bioisosteres,Constrained ligands,Agonism
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