Synthesis and SAR of 4-Aminocyclopentapyrrolidines As N-type Ca2+ Channel Blockers with Analgesic Activity
Xenia Beebe,Daria Darczak,Rodger F. Henry,Timothy Vortherms,Richard Janis,Marian Namovic,Diana Donnelly-Roberts,Karen L. Kage,Carol Surowy,Ivan Milicic,Wende Niforatos,Andrew Swensen,Kennan C. Marsh,Jill M. Wetter,Pamela Franklin,Scott Baker,Chengmin Zhong,Gricelda Simler,Erica Gomez,Janel M. Boyce-Rustay,Chang Z. Zhu,Andrew O. Stewart,Michael F. Jarvis,Victoria E. Scott Bioorganic & Medicinal Chemistry(2012)
关键词
N-type calcium channel,L-type calcium channel,Analgesic activity,SAR,N-tert-Butyl sulfonamide,Enantioselective synthesis
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