Heteroaryl-substituted 4-(1H-pyrazol-1-yl)-5,6-dihydro-1H-pyrrolo[2,3-d]pyrimidine derivatives as potent and selective corticotropin-releasing factor receptor-1 antagonists.
Fabio Maria Sabbatini,Romano Di Fabio,Yves St-Denis,Anna-Maria Capelli,Emiliano Castiglioni,Stefania Contini,Daniele Donati,Elettra Fazzolari,Gabriella Gentile,Fabrizio Micheli,Francesca Pavone,Marilisa Rinaldi,Alessandra Pasquarello,Maria Grazia Zampori,Pina Di Felice,Paola Zarantonello,Roberto Arban,Benedetta Perini,Giovanni Vitulli,Roberto Benedetti,Beatrice Oliosi,Angela Worby CHEMMEDCHEM(2008)
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anxiety,corticotropin releasing factor,CRF1 antagonists,depression
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