Discovery process and characterization of novel carbohydrazide derivatives as potent and selective GHSR1a antagonists.
Fabio Maria Sabbatini,Romano Di Fabio,Mauro Corsi,Paolo Cavanni,Steve M. Bromidge,Yves St-Denis,Lucilla D'Adamo,Stefania Contini,Marilisa Rinaldi,Sebastien Guery,Chiara Savoia,Claudia Mundi,Benedetta Perini,Andrew J. Carpenter,Giovanna Dal Forno,Federico Faggioni,Michela Tessari,Francesca Pavone,Carla Di Francesco,Alberto Buson,Mario Mattioli,Elisabetta Perdona',Sergio Melotto CHEMMEDCHEM(2010)
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antagonists,eating disorders,ghrelin,GHSR1a
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