头孢曲松钠他唑巴坦钠的含量测定
Modern Journal of Integrated Traditional Chinese and Western Medicine(2010)
Abstract
头孢曲松钠为半合成的第3代头孢菌素,对β内酰胺酶稳定.他唑巴坦是β-内酰胺酶抑制剂,能增强抗生素的抗菌活性,又可以扩大其抗菌谱,减少不良反应.酶抑制剂他唑巴坦钠的加入明显提高了头孢曲松钠对耐药菌的抗菌作用,使药理活性较单组分明显增加,且其毒副作用未较原组分增加,有效解决了近年来由于广泛大量选用头孢菌素、导致细菌对第3代头孢菌高度耐药的问题.现将头孢曲松钠他唑巴坦钠的含量测定方法介绍如下.
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