SYNTHESIS OF 1,5-BENZOTHIAZEPINE-1-OXIDE/-1,1-DIOXIDE DERIVATIVES AND 1,2-OXAZIRINO[2,3-a] [1,5] BENZODIAZEPINE
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS(2006)
Abstract
Three 1,3-oxazino[3,2-d][1,5]benzothiazepin-1-one-7-oxide derivatives, three 1,3-oxazino[3,2-d][1,5]benzothiazepin-1-one-7,7-dioxide derivatives, and 1,5-benzothiazepine-1-oxide and 1,5-benzothiazepine-1,1-dioxide derivatives have been synthesized by oxidizing 1,3-oxazino[3,2-d][1,5]benzothiazepin-1-one and 1,5-benzothiazepine with m-chloroperbenzoic acid (MCPBA) as mimetics of benzodiazepinone for studies on relationship of structure and activity, respectively. One 1,2-oxazirino[2,3-a][1,5]benzodiazepine derivative also has been synthesized by the reaction of 1,5-benzodiazepine and m-chloroperbenzoic acid (MCPBA).
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Key words
1,3-oxazino[3,2-d][1,5]benzothiazepin-1-one-7-oxide,1,3-oxazino[3,2-d][1,5]benzothiazepin-1-one-7,7-dioxide,1,5-benzothiazepine-1-oxide,1,5-benzothiazepine-1,1-dioxide,1,2-oxazirino[2,3-a] [1,5]benzodiazepine,oxidation,m-chloroperbenzoic acid
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