Aminocarbonylation route to tolvaptan.
Bioorganic & Medicinal Chemistry Letters（2007）
Abstract
Pd-catalyzed aminocarbonylation between aryl bromide and NH-benzazepinone was effectively carried out to furnish the key intermediate for tolvaptan (up to 85%) in one step.
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Key words
Vasopressin,Palladium,Carbonylation,Cesium salt,DBU
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